تفاعل #746923

ord-0d109a57438c4e769d56ccca9a07b43d

معادلة التفاعل

Cc1ccc(N)cc1Nc1ncc(-c2ccc(C#N)cc2)o1
4-[2-(5-Amino-2-methyl-phenylamino)-oxazol-5-yl]-benzonitrile
CC(=O)Nc1cc([N+](=O)[O-])ccc1C
N-(2-methyl-5-nitro-phenyl)-acetamide
CC(=O)Nc1cc(N)ccc1C
N-(5-Amino-2-methyl-phenyl)-acetamide
Cc1ccc([N+](=O)[O-])cc1Nc1ncc(-c2ccc(C#N)cc2)o1
4-[2-(2-Methyl-5-nitro-phenylamino)-oxazol-5-yl]-benzonitrile
المردود 83.0%

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

الإجراء التجريبي

The same procedure outlined above in the preparation of 4-[2-(5-Amino-2-methyl-phenylamino)-oxazol-5-yl]-benzonitrile was used. However N-(2-methyl-5-nitro-phenyl)-acetamide was used instead N-(5-Amino-2-methyl-phenyl)-acetamide. Yield=83%. m.p.>228° C.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US08080669B2uspto-grants-2011_12