تفاعل #60122

ord-9346bf19280a4b0991d583485fd33fda

معادلة التفاعل

NCCc1ncc(-n2ccnc2)c(-c2ccc(Cl)cc2Cl)n1
4-(2,4-dichlorophenyl)-5-imidazol-1-ylpyrimidin-2-ylethylamine
O=[N+]([O-])c1ccsc1Cl
2-chloro-3-nitrothiophene
COc1nc(NCCNc2ncc(-c3ncc[nH]3)c(-c3ccc(Cl)cc3Cl)n2)ccc1[N+](=O)[O-]
[4-(2,4-dichlorophenyl)-5-imidazol-2-ylpyrimidin-2-yl]{2-[(6-methoxy-5-nitro(2-pyridyl))amino]ethyl}amine
O=[N+]([O-])c1ccsc1NCCNc1ncc(-c2ncc[nH]2)c(-c2ccc(Cl)cc2Cl)n1
[4-(2,4-dichlorophenyl)-5-imidazolylpyrimidin-2-yl]{2-[(3-nitro(2-thienyl))amino]-ethyl}amine

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

الإجراء التجريبي

[4-(2,4-dichlorophenyl)-5-imidazolylpyrimidin-2-yl]{2-[(3-nitro(2-thienyl))amino]-ethyl}amine was prepared from [4-(2,4-dichlorophenyl)-5-imidazol-1-ylpyrimidin-2-ylethylamine and 2-chloro-3-nitrothiophene in accordance with the procedure described above for the preparation of [4-(2,4-dichlorophenyl)-5-imidazol-2-ylpyrimidin-2-yl]{2-[(6-methoxy-5-nitro(2-pyridyl))amino]ethyl}amine.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07425557B2uspto-grants-2008_09