تفاعل #57154

ord-c1e6ba5caf0c4298a22c3b4fc13f826e

معادلة التفاعل

CCn1cc(-c2ccnc3[nH]ccc23)c(-c2ccc(N)cc2)n1
4-[1-ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]aniline
O=C(Cl)C1CCCC1
cyclopentancarbonyl chloride
CCn1cc(-c2ccnc3[nH]ccc23)c(-c2ccc(NC(=O)C3CCCC3)cc2)n1
title compound
CCn1cc(-c2ccnc3[nH]ccc23)c(-c2ccc(NC(=O)C3CCCC3)cc2)n1
N-{4-[1-Ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}cyclopentanecarboxamide

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

الإجراء التجريبي

Following the procedure described in Example 1 with 4-[1-ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]aniline and cyclopentancarbonyl chloride provided the title compound. ESMS [M+H]+: 400.4

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07419988B2uspto-grants-2008_09