تفاعل #56297

ord-5a172908a35746a1ae556a5be665f22e

المذيبات

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

المعالجة

  1. 1
    أخرىviscous residue is obtained
  2. 2
    أخرىThe solid is triturated
  3. 3
    ترشيحcollected by filtration
  4. 4
    غسيلwashed with ether
  5. 5
    تجفيفdried over phosphorus pentoxide

الإجراء التجريبي

7β-(t-Butoxycarbonyl)amino-3-[2-(N-carboethoxysulfamoyl)benzoyloxy]methyl-3-cephem-4-carboxylic acid (2.2 g) is dissolved in ice cooled solution of trifuoroacetic acid (20 ml) and the mixture is stirred for 20 minutes. Then trifluoroacetic acid is taken off under reduced pressure and viscous residue is obtained. The residue becomes solid upon addition of ether (50 ml). The solid is triturated, collected by filtration, washed with ether and dried over phosphorus pentoxide. The procedure provides 7β-amino-3-[2-(N-carboethoxysulfamoyl)benzoyloxy]methyl-3-cephem-4-carboxylic acid (1.55 g).

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US04224441uspto-grants-1980_09