تفاعل #44731

ord-3cef52fa6df843c2bd4ac8e11936d6e9

معادلة التفاعل

Nc1ccc(Oc2ccnc3[nH]ccc23)c(F)c1
3-fluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)aniline
Nc1ccc(Oc2ccnc3[nH]ccc23)c(F)c1
3-Fluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)aniline
Nc1nc(Cl)cc(Cl)n1
4,6-dichloro-2-pyrimidineamine
Nc1nc(Cl)cc(Nc2ccc(Oc3ccnc4[nH]ccc34)c(F)c2)n1
title compound
Nc1nc(Cl)cc(Nc2ccc(Oc3ccnc4[nH]ccc34)c(F)c2)n1
6-Chloro-N4-[3-fluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]pyrimidine-2,4-diamine

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

الإجراء التجريبي

Analogously to example 8, the title compound is synthesized from 266 mg (1.09 mmol) of 3-fluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)aniline (from example XIX) and 179 mg (1.09 mmol) of 4,6-dichloro-2-pyrimidineamine.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07737153B2uspto-grants-2010_06