تفاعل #43811

ord-c0267d7a4d17472887b6e0ded77623d3

المذيبات

ظروف التفاعل

درجة الحرارة
70°CELSIUS
الظروف التفصيلية
See reaction.notes.procedure_details.

المعالجة

  1. 1
    استخلاصextracted with water
  2. 2
    استخلاصextracted with DCM
  3. 3
    غسيلThe organic layer was washed with water
  4. 4
    تركيزconcentrated
  5. 5
    أخرىpurified by preparative LCMS

الإجراء التجريبي

The product of step d.) was dissolved in 3 mL ethanol, treated with 1 M NaOH (500 μL), and heated to 70° C. for one hour. The reaction was diluted in DCM and extracted with water. The aqueous layer was acidified with 1 M HCl and extracted with DCM. The organic layer was washed with water, concentrated and purified by preparative LCMS to give the title compound. MS: ESI (positive): 334 (M+H).

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07732618B2uspto-grants-2010_06