تفاعل #433593

ord-2b018a5bfa7146b2800a231c29e3aeb4

معادلة التفاعل

Nc1ccccc1
Aniline
Nc1ccccc1
aniline
O=[N+]([O-])c1ccc2ncnc(Cl)c2c1
4-chloro-6-nitroquinazoline
O=[N+]([O-])c1ccc2ncnc(Nc3ccccc3)c2c1
4-(phenylamino)-6-nitroquinazoline

الكواشف

لا شيء

المذيبات

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

الإجراء التجريبي

Aniline or derivatized aniline (1 equivalent) is reacted with 4-chloro-6-nitroquinazoline (3.5 equivalents), in a polar solvent such as iso-propyl alcohol. The product, 4-(phenylamino)-6-nitroquinazoline, is obtained after filtration.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07172749B2uspto-grants-2007_02