تفاعل #429216

ord-3f577259a7a748b98a15d36aa6b42723

معادلة التفاعل

ClCCl
methylene chloride
COc1ccc(Sc2nc(-c3ccccc3)n(Cc3cc4c(cc3Cl)OCO4)c2C=O)cc1
product
COc1ccc(Sc2nc(-c3ccccc3)n(Cc3cc4c(cc3Cl)OCO4)c2C=O)cc1
1-((6-chloro-1,3-benzodioxol-5-yl)methyl)-4-((4-methoxyphenyl)thio)-2-phenyl-1H-imidazole-5-carboxaldehyde
[C-]#N.[Na+]
sodium cyanide
CO
methanol
COC(=O)c1c(Sc2ccc(OC)cc2)nc(-c2ccccc2)n1Cc1cc2c(cc1Cl)OCO2
expected product
COC(=O)c1c(Sc2ccc(OC)cc2)nc(-c2ccccc2)n1Cc1cc2c(cc1Cl)OCO2
methyl 1-((6-chloro-1,3-benzodioxol-5-yl)methyl)-4-((4-methoxyphenyl)thio)-2-phenyl-1H-imidazole-5-carboxylate

المذيبات

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

الإجراء التجريبي

The operation is carried out as in Example 9 starting with 2 g of the product of Example 20 using 10 g of manganese oxide, 1 g of sodium cyanide, 200 ml of methanol, 40 ml of methylene chloride and 600 ul of acetic acid, in this way 1.64 g of expected product is obtained (M.p.=161° C.).

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US05856509uspto-grants-1999_01