تفاعل #42753

ord-eb3fa833e9984931ac0a2ad081535a12

المذيبات

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

المعالجة

  1. 1
    استخلاصthe mixture is extracted with ethyl acetate (3×200 ml)
  2. 2
    تجفيفdried (MgSO4)
  3. 3
    ترشيحfiltered
  4. 4
    تركيزconcentrated
  5. 5
    أخرىto afford a yellow suspension
  6. 6
    أخرىThe suspension is triturated with hexanes

الإجراء التجريبي

A solution of 7-(benzhydrylideneamino)-3-(4-chlorophenyl)-2-isopropyl-chromen-4-one (5.72 g, 12 mmol) in tetrahydrofuran (150 ml) is treated with 2M HCl solution (150 ml) and allowed to stir at room temperature for 1 hour. The solution is basified with 17% ammonia solution (150 ml), and the mixture is extracted with ethyl acetate (3×200 ml). The organic extracts are combined, dried (MgSO4), filtered and concentrated to afford a yellow suspension. The suspension is triturated with hexanes to afford the title compound as a pale yellow solid, which is isolated by filtration and dried in vacuo overnight.

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07732435B2uspto-grants-2010_06