تفاعل #40823

ord-25cfcf96b25d4fc6b54c9b584a00826c

معادلة التفاعل

CCOC(=O)c1ccc(-c2ccc(C(F)(F)F)cc2)c(-c2ccccc2)n1
ethyl 5-(4-trifluoromethylphenyl)-6-phenylpyridine-2-carboxylate
CCOC(=O)c1ccc(-c2ccc(C(F)(F)F)cc2)c(-c2ccccc2)n1
ethyl 6-phenyl-5-(4-trifluoromethylphenyl)-pyridine-2-carboxylate
CCOC(=O)c1ccc(-c2ccc(C(F)(F)F)cc2)c(-c2ccccc2)n1
Compound 25
CCOC(=O)c1ccc(-c2ccc(C(F)(F)F)cc2)c(-c2ccccc2)n1
ethyl 6-phenyl-5-(4-trifluoromethylphenyl)-pyridine-2-carboxylate
CC(C)[CH2][AlH][CH2]C(C)C
DIBAL-H
O=Cc1ccc(-c2ccc(C(F)(F)F)cc2)c(-c2ccccc2)n1
title compound
O=Cc1ccc(-c2ccc(C(F)(F)F)cc2)c(-c2ccccc2)n1
5-(4-Trifluoromethylphenyl)-6-phenylpyridine-2-carbaldehyde

المذيبات

ظروف التفاعل

الظروف التفصيلية
See reaction.notes.procedure_details.

المعالجة

  1. 1
    أخرىwere reacted

الإجراء التجريبي

Following General Procedure L, ethyl 5-(4-trifluoromethylphenyl)-6-phenylpyridine-2-carboxylate (Compound 25, 74 mg, 0.20 mmol) and DIBAL-H (0.3 ml, 0.30 mmol, 1.0 M in hexane) in CH2Cl2 (3 ml) were reacted to produce the title compound after purification by column chromatography (silica gel, 15% ethyl acetate in hexane).

المصدر

DOI: 10.6084/m9.figshare.5104873.v1براءة الاختراع: US07728014B2uspto-grants-2010_06