تفاعل #1782778

معادلة التفاعل

rac-N2-(7-methoxy-indan-1-yl)-4H-benzo[d][1,3]oxazine-2,6-diamine

rac-N2-(7-Methoxy-indan-1-yl)-4H-benzo[d][1,3]oxazine-2,6-diamine

methoxyacetyl chloride

→

title compound

المردود 61.0%

rac-2-Methoxy-N-[2-(7-methoxy-indan-1-ylamino)-4H-benzo[d][1,3]oxazin-6-yl]-acetamide

المردود 61.0%

ظروف التفاعل

الإجراء التجريبي

Prepared from rac-N2-(7-methoxy-indan-1-yl)-4H-benzo[d][1,3]oxazine-2,6-diamine (Example 10) (100 mg, 0.323 mmol) and methoxyacetyl chloride (32 ul, 0.356 mmol) according to the procedure described for Example 17. Obtained the title compound as a white solid (75 mg, 61%), MS (ISP) m/e=382.2 [(M+H)+].

المصدر