بحث البنية الفرعية

176883

CC1(C)OC[C@@H](Cn2ccc([N+](=O)[O-])n2)O1
Reaction #47262
1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-3-nitro-1H-pyrazole
المردود 73.0%DOI: 10.6084/m9.figshare.5104873.v1
CC1(C)OC[C@@H](Cn2ccc(N)n2)O1
Reaction #47263
1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-ylamine
المردود 98.5%DOI: 10.6084/m9.figshare.5104873.v1
O=C(Nc1ccn(C[C@@H](O)CO)n1)[C@H](CC1CCCCC1)N1CC(Oc2ccccc2Cl)=CC1=O
Reaction #47272
(S)-2-[4-(2-chloro-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-3-cyclohexyl-N-[1-((R)-2,3-dihydroxy-propyl)-1-H-pyrazol-3-yl]-propionamide
المردود 83.0%DOI: 10.6084/m9.figshare.5104873.v1
CC1(C)OC[C@@H](Cn2ccc(N3C(=O)c4ccccc4C3=O)n2)O1
Reaction #47279
2-[1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-yl]-isoindole-1,3-dione
المردود 74.1%DOI: 10.6084/m9.figshare.5104873.v1
CC1(C)OC[C@@H](Cn2ccc(N)n2)O1
Reaction #47280
1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-ylamine
المردود 94.6%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H](O)CO)n1)N1CC(Oc2ccccc2Cl)=CC1=O
Reaction #47281
(S)-2-[4-(2-chloro-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-4-methyl-pentanoic acid [1-((R)-2,3-dihydroxy-propyl)-1H-pyrazol-3-yl]-amide
المردود 96.7%DOI: 10.6084/m9.figshare.5104873.v1
CC1(C)OC[C@@H](Cn2ccc([N+](=O)[O-])n2)O1
Reaction #47294
1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-3-nitro-1H-pyrazole
المردود 72.0%DOI: 10.6084/m9.figshare.5104873.v1
CC1(C)OC[C@@H](Cn2ccc(N)n2)O1
Reaction #47295
1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-ylamine
المردود 98.5%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H](O)CO)n1)N1CC(Oc2cccc(Cl)c2Cl)=CC1=O
Reaction #47296
(S)-2-[4-(2,3-dichloro-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-4-methyl-pentanoic acid [1-((R)-2,3-dihydroxy-propyl)-1H-pyrazol-3-yl]-amide
DOI: 10.6084/m9.figshare.5104873.v1
CCOc1ccccc1OC1=CC(=O)N([C@@H](CC(C)C)C(=O)Nc2ccn(C[C@@H](O)CO)n2)C1
Reaction #47299
(S)-2-[4-(2-ethoxy-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-4-methyl-pentanoic acid [1-((R)-2,3-dihydroxy-propyl)-1H-pyrazol-3-yl]-amide
DOI: 10.6084/m9.figshare.5104873.v1
O=C(Nc1ccn(C[C@@H](O)CO)n1)[C@H](CC1CCCC1)N1CC(Oc2c(F)cccc2F)=CC1=O
Reaction #47301
(S)-3-cyclopentyl-2-[4-(2,6-difluoro-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-N-[1-((R)-2,3-dihydroxy-propyl)-1H-pyrazol-3-yl]-propionamide
المردود 64.9%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H]2COC(C)(C)O2)n1)N1CC(Oc2cccc(C(F)(F)F)c2)=CC1=O
Reaction #47329
(S)-4-methyl-2-[2-oxo-4-(3-trifluoromethyl-phenoxy)-2,5-dihydro-pyrrol-1-yl]-pentanoic acid [1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-yl]-amide
المردود 51.0%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H](O)CO)n1)N1CC(Oc2cccc(C(F)(F)F)c2)=CC1=O
Reaction #47330
(S)-4-methyl-2-[2-oxo-4-(3-trifluoromethyl-phenoxy)-2,5-dihydro-pyrrol-1-yl]-pentanoic acid [1-((R)-2,3-dihydroxy-propyl)-1H-pyrazol-3-yl]-amide
المردود 78.0%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H]2COC(C)(C)O2)n1)N1CC(Oc2cccc(Cl)c2F)=CC1=O
Reaction #47335
(S)-2-[4-(3-chloro-2-fluoro-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-4-methyl-pentanoic acid [1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-yl]-amide
المردود 49.0%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H](O)CO)n1)N1CC(Oc2cccc(Cl)c2F)=CC1=O
Reaction #47336
(S)-2-[4-(3-chloro-2-fluoro-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-4-methyl-pentanoic acid [1-((R)-2,3-dihydroxy-propyl)-1H-pyrazol-3-yl]-amide
المردود 79.0%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H]2COC(C)(C)O2)n1)N1CC(Oc2cccc3c2CCCC3)=CC1=O
Reaction #47341
(S)-4-methyl-2-[2-oxo-4-(5,6,7,8-tetrahydro-naphthalen-1-yloxy)-2,5-dihydro-pyrrol-1-yl]-pentanoic acid [1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-yl]-amide
المردود 48.4%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H](O)CO)n1)N1CC(Oc2cccc3c2CCCC3)=CC1=O
Reaction #47342
(S)-4-methyl-2-[2-oxo-4-(5,6,7,8-tetrahydro-naphthalen-1-yloxy)-2,5-dihydro-pyrrol-1-yl]-pentanoic acid [1-((R)-2,3-dihydroxy-propyl)-1H-pyrazol-3-yl]-amide
المردود 72.5%DOI: 10.6084/m9.figshare.5104873.v1
COc1ccc(OC2=CC(=O)N([C@@H](CC(C)C)C(=O)Nc3ccn(C[C@@H]4COC(C)(C)O4)n3)C2)cc1
Reaction #47348
(S)-2-[4-(4-methoxy-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-4-methyl-pentanoic acid [1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-yl]-amide
المردود 68.0%DOI: 10.6084/m9.figshare.5104873.v1
COc1ccc(OC2=CC(=O)N([C@@H](CC(C)C)C(=O)Nc3ccn(C[C@@H](O)CO)n3)C2)cc1
Reaction #47349
(S)-2-[4-(4-methoxy-phenoxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-4-methyl-pentanoic acid [1-((R)-2,3-dihydroxy-propyl)-1H-pyrazol-3-yl]-amide
المردود 86.1%DOI: 10.6084/m9.figshare.5104873.v1
CC(C)C[C@@H](C(=O)Nc1ccn(C[C@@H]2COC(C)(C)O2)n1)N1CC(Oc2cccc3ccccc23)=CC1=O
Reaction #47354
(S)-4-methyl-2-[4-(naphthalen-1-yloxy)-2-oxo-2,5-dihydro-pyrrol-1-yl]-pentanoic acid [1-((R)-2,2-dimethyl-[1,3]dioxolan-4-yl-methyl)-1H-pyrazol-3-yl]-amide
المردود 76.0%DOI: 10.6084/m9.figshare.5104873.v1
الصفحة 1التالي