بحث البنية الفرعية

136

Cc1cccnc1N[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #656
المردود 69.8%
Cc1cccnc1N[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #657
المردود 82.4%
Cc1cccnc1N[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #675539
title compound
المردود 60.0%DOI: 10.6084/m9.figshare.5104873.v1
Cc1cccnc1N(C(=O)c1ccc(Br)cc1)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #675550
title compound
المردود 50.0%DOI: 10.6084/m9.figshare.5104873.v1
Cc1ccc[n+]([O-])c1N[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #675553
title compound
المردود 25.0%DOI: 10.6084/m9.figshare.5104873.v1
Cc1cccnc1N(C(=O)c1ccc(-c2cnn(C)c2-c2nn[nH]n2)cc1)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #675564
tert-butyl (3R)-3-(4-(1-methyl-5-(2H-tetrazol-5-yl)-1H-pyrazol-4-yl)-N-(3-methylpyridin-2-yl)benzamido)piperidine-1-carboxylate
المردود 90.5%DOI: 10.6084/m9.figshare.5104873.v1
Cc1cccnc1N(C(=O)c1ccc(-c2cnn(C)c2C#N)cc1)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #675565
tert-butyl (3R)-3-{[4-(5-cyano-1-methyl-1H-pyrazol-4-yl)benzoyl](3-methylpyridin-2-yl)amino}piperidine-1-carboxylate
المردود 73.0%DOI: 10.6084/m9.figshare.5104873.v1
CCOC(=O)O[C@@H](C)n1nnc(-c2c(-c3ccc(C(=O)N(c4ncccc4C)[C@@H]4CCCN(C(=O)OC(C)(C)C)C4)cc3)cnn2C)n1
Reaction #675566
tert-butyl (3R)-3-[{4-[5-(2-{(1S)-1-[(ethoxycarbonyl)oxy]ethyl}-2H-tetrazol-5-yl)-1-methyl-1H-pyrazol-4-yl]benzoyl}(3-methylpyridin-2-yl)amino]piperidine-1-carboxylate
المردود 77.0%DOI: 10.6084/m9.figshare.5104873.v1
Cc1cccnc1N(C(=O)c1ccc(-c2cnn(C)c2C(=O)O)cc1)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #675567
4-(4-{[(3R)-1-(tert-butoxycarbonyl)piperidin-3-yl](3-methylpyridin-2-yl)carbamoyl}phenyl)-1-methyl-1H-pyrazole-5-carboxylic acid
المردود 261.0%DOI: 10.6084/m9.figshare.5104873.v1
Cc1ccc[n+]([O-])c1N(C(=O)c1ccc(-c2cnn3cccnc23)cc1)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #675568
(R)-2-(N-(1-(tert-butoxycarbonyl)piperidin-3-yl)-4-(pyrazolo[1,5-a]pyrimidin-3-yl)benzamido)-3-methylpyridine 1-oxide
DOI: 10.6084/m9.figshare.5104873.v1
Cc1cccnc1N(C(=O)c1ccc(-c2cnn3cccnc23)cc1)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1
Reaction #675569
title compound
DOI: 10.6084/m9.figshare.5104873.v1
Cc1cccnc1N(C(=O)c1ccc(-c2cnn3cccnc23)cc1)[C@@H]1CCCNC1.Cl
Reaction #675570
N-(3-methylpyridin-2-yl)-N-[(3R)-piperidin-3-yl]-4-(pyrazolo[1,5-a]pyrimidin-3-yl)benzamide hydrochloride
DOI: 10.6084/m9.figshare.5104873.v1
COC(=O)c1c(-c2ccc(C(=O)N(c3ncccc3C)[C@@H]3CCCN(C(=O)OC(C)(C)C)C3)cc2)cnn1C
Reaction #675578
desired title compound
المردود 94.5%DOI: 10.6084/m9.figshare.5104873.v1
Cc1cccnc1N(C(=O)c1ccc(-c2cnn(C)c2-c2nn[nH]n2)cc1)[C@@H]1CCCNC1
Reaction #675580
N-(3-methylpyridin-2-yl)-4-[1-methyl-5-(2H-tetrazol-5-yl)-1H-pyrazol-4-yl]-N-[(3R)-piperidin-3-yl]benzamide
المردود 108.8%DOI: 10.6084/m9.figshare.5104873.v1
CCOC(=O)OC(C)n1c(-c2c(-c3ccc(C(=O)N(c4ncccc4C)[C@@H]4CCCNC4)cc3)cnn2C)noc1=O
Reaction #675581
ethyl 1-{3-[1-methyl-4-(4-{(3-methylpyridin-2-yl)[(3R)-piperidin-3-yl]carbamoyl}phenyl)-1H-pyrazol-5-yl]-5-oxo-1,2,4-oxadiazol-4(5H)-yl}ethyl carbonate
المردود 86.9%DOI: 10.6084/m9.figshare.5104873.v1
CCOC(=O)O[C@@H](C)n1nnc(-c2c(-c3ccc(C(=O)N(c4ncccc4C)[C@@H]4CCCNC4)cc3)cnn2C)n1
Reaction #675582
ethyl (1S)-1-{5-[1-methyl-4-(4-{(3-methylpyridin-2-yl)[(3R)-piperidin-3-yl]carbamoyl}phenyl)-1H-pyrazol-5-yl]-2H-tetrazol-2-yl}ethyl carbonate
المردود 65.1%DOI: 10.6084/m9.figshare.5104873.v1
CCOC(=O)O[C@H](C)n1nnc(-c2c(-c3ccc(C(=O)N(c4ncccc4C)[C@@H]4CCCN(C(=O)OC(C)(C)C)C4)cc3)cnn2C)n1
Reaction #2103821
DOI: 10.1038/s41557
CCOC(=O)O[C@H](C)n1nnc(-c2c(-c3ccc(C(=O)N(c4ncccc4C)[C@@H]4CCCN(C(=O)OC(C)(C)C)C4)cc3)cnn2C)n1
Reaction #2103822
DOI: 10.1038/s41557
CCOC(=O)O[C@H](C)n1nnc(-c2c(-c3ccc(C(=O)N(c4ncccc4C)[C@@H]4CCCN(C(=O)OC(C)(C)C)C4)cc3)cnn2C)n1
Reaction #2103823
DOI: 10.1038/s41557
CCOC(=O)O[C@H](C)n1nnc(-c2c(-c3ccc(C(=O)N(c4ncccc4C)[C@@H]4CCCN(C(=O)OC(C)(C)C)C4)cc3)cnn2C)n1
Reaction #2103824
DOI: 10.1038/s41557
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